Multicomponent Pharmaceutical Solids

Multicomponent pharmaceutical materials are solids in which at least one component is an active pharmaceutical ingredient (API). This kind of pharmaceutical solid has attracted interest in the past decade as a promising alternative to the laborious and expensive process of traditional pipeline drug...

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collection Directory of Open Access Books
description Multicomponent pharmaceutical materials are solids in which at least one component is an active pharmaceutical ingredient (API). This kind of pharmaceutical solid has attracted interest in the past decade as a promising alternative to the laborious and expensive process of traditional pipeline drug development. The application of crystal engineering techniques into the design of pharmaceutical salts, co-crystals, and other multicomponent materials, in addition to the achievement of more environmentally friendly synthetic approaches, has succeeded in modulating the physicochemical, mechanical, and pharmacokinetic properties of drugs, thereby working toward the enhancement of their clinical performance. This Special Issue welcomed original research articles and reviews devoted to all aspects related to the field of multicomponent pharmaceutical solids. Our interests include the fundamentals of applied research, using theoretical and experimental approaches, the development of synthetic methods, the screening of multicomponent materials, structure–activity rationale, the salt–co-crystal continuum identification, the enhancement in physicochemical/mechanical/pharmacokinetic performance, as well as the functionality and applications of multicomponent pharmaceuticals solids.
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language eng
publishDate 2023
publishDateRange 2023
publishDateSort 2023
publisher MDPI - Multidisciplinary Digital Publishing Institute
publisherStr MDPI - Multidisciplinary Digital Publishing Institute
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spelling doab-20.500.12854ir-1000632024-03-28T03:32:40Z Multicomponent Pharmaceutical Solids Choquesillo-Lazarte, Duane Dominguez-Martin, Alicia solvate polymorph bilastine crystal structure determination single crystal X-ray diffraction structure determination from powder diffraction aripiprazole multicomponent crystal crystal structure solubility drug–drug cocrystal furosemide ethenzamide piroxicam mechanochemical synthesis amorphous drug characterization methods crystallization physical stability molecular mobility aminoglutethimide eutectic mixture melt phase diagram nucleobases multicomponent solids crystal engineering DFT H-bonding pyridinecarboxamides cocrystals mandelic acid X-ray structure DFT calculations xanthines theophylline squaric acid controlled release dissolution lidocaine mechanochemistry multicomponent materials API pharmaceutical solids diclofenac pharmaceutical solid forms n/a thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general thema EDItEUR::P Mathematics and Science::PH Physics Multicomponent pharmaceutical materials are solids in which at least one component is an active pharmaceutical ingredient (API). This kind of pharmaceutical solid has attracted interest in the past decade as a promising alternative to the laborious and expensive process of traditional pipeline drug development. The application of crystal engineering techniques into the design of pharmaceutical salts, co-crystals, and other multicomponent materials, in addition to the achievement of more environmentally friendly synthetic approaches, has succeeded in modulating the physicochemical, mechanical, and pharmacokinetic properties of drugs, thereby working toward the enhancement of their clinical performance. This Special Issue welcomed original research articles and reviews devoted to all aspects related to the field of multicomponent pharmaceutical solids. Our interests include the fundamentals of applied research, using theoretical and experimental approaches, the development of synthetic methods, the screening of multicomponent materials, structure–activity rationale, the salt–co-crystal continuum identification, the enhancement in physicochemical/mechanical/pharmacokinetic performance, as well as the functionality and applications of multicomponent pharmaceuticals solids. 2023-05-11T17:18:59Z 2023-05-11T17:18:59Z 2023 book ONIX_20230511_9783036572161_80 9783036572161 9783036572178 https://directory.doabooks.org/handle/20.500.12854/100063 eng image/jpeg Attribution 4.0 International https://mdpi.com/books/pdfview/book/7156 https://mdpi.com/books/pdfview/book/7156 MDPI - Multidisciplinary Digital Publishing Institute 10.3390/books978-3-0365-7217-8 10.3390/books978-3-0365-7217-8 46cabcaa-dd94-4bfe-87b4-55023c1b36d0 9783036572161 9783036572178 178 Basel open access
spellingShingle solvate
polymorph
bilastine
crystal structure determination
single crystal X-ray diffraction
structure determination from powder diffraction
aripiprazole
multicomponent crystal
crystal structure
solubility
drug–drug cocrystal
furosemide
ethenzamide
piroxicam
mechanochemical synthesis
amorphous drug
characterization methods
crystallization
physical stability
molecular mobility
aminoglutethimide
eutectic mixture
melt phase diagram
nucleobases
multicomponent solids
crystal engineering
DFT
H-bonding
pyridinecarboxamides
cocrystals
mandelic acid
X-ray structure
DFT calculations
xanthines
theophylline
squaric acid
controlled release
dissolution
lidocaine
mechanochemistry
multicomponent materials
API
pharmaceutical solids
diclofenac
pharmaceutical solid forms
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PH Physics
Multicomponent Pharmaceutical Solids
title Multicomponent Pharmaceutical Solids
title_full Multicomponent Pharmaceutical Solids
title_fullStr Multicomponent Pharmaceutical Solids
title_full_unstemmed Multicomponent Pharmaceutical Solids
title_short Multicomponent Pharmaceutical Solids
title_sort multicomponent pharmaceutical solids
topic solvate
polymorph
bilastine
crystal structure determination
single crystal X-ray diffraction
structure determination from powder diffraction
aripiprazole
multicomponent crystal
crystal structure
solubility
drug–drug cocrystal
furosemide
ethenzamide
piroxicam
mechanochemical synthesis
amorphous drug
characterization methods
crystallization
physical stability
molecular mobility
aminoglutethimide
eutectic mixture
melt phase diagram
nucleobases
multicomponent solids
crystal engineering
DFT
H-bonding
pyridinecarboxamides
cocrystals
mandelic acid
X-ray structure
DFT calculations
xanthines
theophylline
squaric acid
controlled release
dissolution
lidocaine
mechanochemistry
multicomponent materials
API
pharmaceutical solids
diclofenac
pharmaceutical solid forms
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PH Physics
topic_facet solvate
polymorph
bilastine
crystal structure determination
single crystal X-ray diffraction
structure determination from powder diffraction
aripiprazole
multicomponent crystal
crystal structure
solubility
drug–drug cocrystal
furosemide
ethenzamide
piroxicam
mechanochemical synthesis
amorphous drug
characterization methods
crystallization
physical stability
molecular mobility
aminoglutethimide
eutectic mixture
melt phase diagram
nucleobases
multicomponent solids
crystal engineering
DFT
H-bonding
pyridinecarboxamides
cocrystals
mandelic acid
X-ray structure
DFT calculations
xanthines
theophylline
squaric acid
controlled release
dissolution
lidocaine
mechanochemistry
multicomponent materials
API
pharmaceutical solids
diclofenac
pharmaceutical solid forms
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PH Physics
url ONIX_20230511_9783036572161_80