Synthesis of Heteroaromatic Compounds

This Special Issue, entitled the “Synthesis of Heteroaromatic Compounds”, is an outstanding collection of fourteen original research papers and six review articles that discuss the advances made in both conventional and green preparatory methods, as well as the properties and applications of heteroa...

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description This Special Issue, entitled the “Synthesis of Heteroaromatic Compounds”, is an outstanding collection of fourteen original research papers and six review articles that discuss the advances made in both conventional and green preparatory methods, as well as the properties and applications of heteroaromatic molecules in industrial and medicinal chemistry areas of study.The collected works featured herein collate contributions from a truly international and diverse array of ninety experts in the fields of heteroaromatic compound synthesis, QSAR studies, computational chemistry and molecular docking, as well as bioactivity studies.
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institution Directory of Open Access Books
language eng
publishDate 2023
publishDateRange 2023
publishDateSort 2023
publisher MDPI - Multidisciplinary Digital Publishing Institute
publisherStr MDPI - Multidisciplinary Digital Publishing Institute
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spelling doab-20.500.12854ir-1008132024-03-28T03:33:07Z Synthesis of Heteroaromatic Compounds Sloop, Joseph heteroaromatics C-H bond functionalization oxidative cyclization cross-coupling amination triazoles palladium carbene ligands heterocycles nitrogen-containing heterocycles synthesis antiviral agents viruses COVID-19 inhibition Mpro inhibitors drug design and synthesis structure-activity relationships (SAR) s-tetrazine 4H-1,2,4-triazole pinner reaction 1,2,3-triazole fused 1,2,3-triazole 1,2,3-triazolo[4,5-b]pyrazine 1,2,3-triazolo[4,5-c]pyridazine 1,2,3-triazolo[4,5-d]pyridazine 1,2,3-triazolo[1,5-a]pyrazine 1,2,3-triazolo[1,5-b]pyridazine triazolopyrazine triazolopyridazine practical applications spiro π-conjugated compound chiral compound thiophene furan pyrrole nucleophilic aromatic substitution circular dichroism circularly polarized luminescence pyridines 1,3,4-thiadiazoles 1,3-thiazoles hydrazonoyl halides molecular docking anticancer activity 1,3,4-oxadiazoles organic ligands substitution diisopropyl iminodiacetate pyrimidine benzimidazole aza-Diels–Alder reaction Povarov reaction oxidation fluorescence aggregation-induced emission mechanochromic properties heterocycle natural product nicotinic acid fungicidal activity 4-pyrone DMF-DMA enamination cycloaddition merocyanine 1,6-conjugate addition solvatochromism fluorophore acetylcoumarin thiazoles VEGFR-2 polyfluoroflavones 1H-1,2,4-triazole imidazole regioselectivity azolyl-substituted flavones photoluminescence 4-pyridone oxazinone ring-opening aldehyde-lactol tautomerism ammonium acetate diazirine medicinal chemistry photoaffinity labeling metathesis carboaromatics 4,5-dihydro-5-oxo-pyrazolo[1,5-a]thieno[2,3-c]pyrimidines novel scaffold molecular dynamic studies proximity frequencies (PF) GABAA receptor subtype GABAA receptor ligands antibacterial anticancer antifibrotic antifungal antimicrobial antiviral appel salt 1,2,3-dithiazole disulfide bridge herbicidal chalcone heteroaromatic hybrid chalcone n/a thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general thema EDItEUR::P Mathematics and Science::PN Chemistry thema EDItEUR::P Mathematics and Science::PN Chemistry::PNN Organic chemistry This Special Issue, entitled the “Synthesis of Heteroaromatic Compounds”, is an outstanding collection of fourteen original research papers and six review articles that discuss the advances made in both conventional and green preparatory methods, as well as the properties and applications of heteroaromatic molecules in industrial and medicinal chemistry areas of study.The collected works featured herein collate contributions from a truly international and diverse array of ninety experts in the fields of heteroaromatic compound synthesis, QSAR studies, computational chemistry and molecular docking, as well as bioactivity studies. 2023-06-23T09:44:45Z 2023-06-23T09:44:45Z 2023 book ONIX_20230623_9783036575636_45 9783036575636 9783036575629 https://directory.doabooks.org/handle/20.500.12854/100813 eng image/jpeg Attribution 4.0 International https://mdpi.com/books/pdfview/book/7276 https://mdpi.com/books/pdfview/book/7276 MDPI - Multidisciplinary Digital Publishing Institute 10.3390/books978-3-0365-7562-9 10.3390/books978-3-0365-7562-9 46cabcaa-dd94-4bfe-87b4-55023c1b36d0 9783036575636 9783036575629 446 Basel open access
spellingShingle heteroaromatics
C-H bond functionalization
oxidative cyclization
cross-coupling
amination
triazoles
palladium
carbene ligands
heterocycles
nitrogen-containing heterocycles
synthesis
antiviral agents
viruses
COVID-19
inhibition
Mpro inhibitors
drug design and synthesis
structure-activity relationships (SAR)
s-tetrazine
4H-1,2,4-triazole
pinner reaction
1,2,3-triazole
fused 1,2,3-triazole
1,2,3-triazolo[4,5-b]pyrazine
1,2,3-triazolo[4,5-c]pyridazine
1,2,3-triazolo[4,5-d]pyridazine
1,2,3-triazolo[1,5-a]pyrazine
1,2,3-triazolo[1,5-b]pyridazine
triazolopyrazine
triazolopyridazine
practical applications
spiro π-conjugated compound
chiral compound
thiophene
furan
pyrrole
nucleophilic aromatic substitution
circular dichroism
circularly polarized luminescence
pyridines
1,3,4-thiadiazoles
1,3-thiazoles
hydrazonoyl halides
molecular docking
anticancer activity
1,3,4-oxadiazoles
organic ligands
substitution
diisopropyl iminodiacetate
pyrimidine
benzimidazole
aza-Diels–Alder reaction
Povarov reaction
oxidation
fluorescence
aggregation-induced emission
mechanochromic properties
heterocycle
natural product
nicotinic acid
fungicidal activity
4-pyrone
DMF-DMA
enamination
cycloaddition
merocyanine
1,6-conjugate addition
solvatochromism
fluorophore
acetylcoumarin
thiazoles
VEGFR-2
polyfluoroflavones
1H-1,2,4-triazole
imidazole
regioselectivity
azolyl-substituted flavones
photoluminescence
4-pyridone
oxazinone
ring-opening
aldehyde-lactol tautomerism
ammonium acetate
diazirine
medicinal chemistry
photoaffinity labeling
metathesis
carboaromatics
4,5-dihydro-5-oxo-pyrazolo[1,5-a]thieno[2,3-c]pyrimidines
novel scaffold
molecular dynamic studies
proximity frequencies (PF)
GABAA receptor subtype
GABAA receptor ligands
antibacterial
anticancer
antifibrotic
antifungal
antimicrobial
antiviral
appel salt
1,2,3-dithiazole
disulfide bridge
herbicidal
chalcone
heteroaromatic
hybrid chalcone
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
thema EDItEUR::P Mathematics and Science::PN Chemistry::PNN Organic chemistry
Synthesis of Heteroaromatic Compounds
title Synthesis of Heteroaromatic Compounds
title_full Synthesis of Heteroaromatic Compounds
title_fullStr Synthesis of Heteroaromatic Compounds
title_full_unstemmed Synthesis of Heteroaromatic Compounds
title_short Synthesis of Heteroaromatic Compounds
title_sort synthesis of heteroaromatic compounds
topic heteroaromatics
C-H bond functionalization
oxidative cyclization
cross-coupling
amination
triazoles
palladium
carbene ligands
heterocycles
nitrogen-containing heterocycles
synthesis
antiviral agents
viruses
COVID-19
inhibition
Mpro inhibitors
drug design and synthesis
structure-activity relationships (SAR)
s-tetrazine
4H-1,2,4-triazole
pinner reaction
1,2,3-triazole
fused 1,2,3-triazole
1,2,3-triazolo[4,5-b]pyrazine
1,2,3-triazolo[4,5-c]pyridazine
1,2,3-triazolo[4,5-d]pyridazine
1,2,3-triazolo[1,5-a]pyrazine
1,2,3-triazolo[1,5-b]pyridazine
triazolopyrazine
triazolopyridazine
practical applications
spiro π-conjugated compound
chiral compound
thiophene
furan
pyrrole
nucleophilic aromatic substitution
circular dichroism
circularly polarized luminescence
pyridines
1,3,4-thiadiazoles
1,3-thiazoles
hydrazonoyl halides
molecular docking
anticancer activity
1,3,4-oxadiazoles
organic ligands
substitution
diisopropyl iminodiacetate
pyrimidine
benzimidazole
aza-Diels–Alder reaction
Povarov reaction
oxidation
fluorescence
aggregation-induced emission
mechanochromic properties
heterocycle
natural product
nicotinic acid
fungicidal activity
4-pyrone
DMF-DMA
enamination
cycloaddition
merocyanine
1,6-conjugate addition
solvatochromism
fluorophore
acetylcoumarin
thiazoles
VEGFR-2
polyfluoroflavones
1H-1,2,4-triazole
imidazole
regioselectivity
azolyl-substituted flavones
photoluminescence
4-pyridone
oxazinone
ring-opening
aldehyde-lactol tautomerism
ammonium acetate
diazirine
medicinal chemistry
photoaffinity labeling
metathesis
carboaromatics
4,5-dihydro-5-oxo-pyrazolo[1,5-a]thieno[2,3-c]pyrimidines
novel scaffold
molecular dynamic studies
proximity frequencies (PF)
GABAA receptor subtype
GABAA receptor ligands
antibacterial
anticancer
antifibrotic
antifungal
antimicrobial
antiviral
appel salt
1,2,3-dithiazole
disulfide bridge
herbicidal
chalcone
heteroaromatic
hybrid chalcone
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
thema EDItEUR::P Mathematics and Science::PN Chemistry::PNN Organic chemistry
topic_facet heteroaromatics
C-H bond functionalization
oxidative cyclization
cross-coupling
amination
triazoles
palladium
carbene ligands
heterocycles
nitrogen-containing heterocycles
synthesis
antiviral agents
viruses
COVID-19
inhibition
Mpro inhibitors
drug design and synthesis
structure-activity relationships (SAR)
s-tetrazine
4H-1,2,4-triazole
pinner reaction
1,2,3-triazole
fused 1,2,3-triazole
1,2,3-triazolo[4,5-b]pyrazine
1,2,3-triazolo[4,5-c]pyridazine
1,2,3-triazolo[4,5-d]pyridazine
1,2,3-triazolo[1,5-a]pyrazine
1,2,3-triazolo[1,5-b]pyridazine
triazolopyrazine
triazolopyridazine
practical applications
spiro π-conjugated compound
chiral compound
thiophene
furan
pyrrole
nucleophilic aromatic substitution
circular dichroism
circularly polarized luminescence
pyridines
1,3,4-thiadiazoles
1,3-thiazoles
hydrazonoyl halides
molecular docking
anticancer activity
1,3,4-oxadiazoles
organic ligands
substitution
diisopropyl iminodiacetate
pyrimidine
benzimidazole
aza-Diels–Alder reaction
Povarov reaction
oxidation
fluorescence
aggregation-induced emission
mechanochromic properties
heterocycle
natural product
nicotinic acid
fungicidal activity
4-pyrone
DMF-DMA
enamination
cycloaddition
merocyanine
1,6-conjugate addition
solvatochromism
fluorophore
acetylcoumarin
thiazoles
VEGFR-2
polyfluoroflavones
1H-1,2,4-triazole
imidazole
regioselectivity
azolyl-substituted flavones
photoluminescence
4-pyridone
oxazinone
ring-opening
aldehyde-lactol tautomerism
ammonium acetate
diazirine
medicinal chemistry
photoaffinity labeling
metathesis
carboaromatics
4,5-dihydro-5-oxo-pyrazolo[1,5-a]thieno[2,3-c]pyrimidines
novel scaffold
molecular dynamic studies
proximity frequencies (PF)
GABAA receptor subtype
GABAA receptor ligands
antibacterial
anticancer
antifibrotic
antifungal
antimicrobial
antiviral
appel salt
1,2,3-dithiazole
disulfide bridge
herbicidal
chalcone
heteroaromatic
hybrid chalcone
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
thema EDItEUR::P Mathematics and Science::PN Chemistry::PNN Organic chemistry
url ONIX_20230623_9783036575636_45