Molecular Methods in Antibiotics Discovery

This Special Issue welcomed manuscripts that describe new compounds with antibiotic activity. Eleven papers were published, most of which describe novel compounds, including homopolymers, cyclic imides, antimicrobial peptides, nucleic acids, and derivatives of quinone, benzamidine, thiazole, and pyr...

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Jazyk:angličtina
Vydáno: MDPI - Multidisciplinary Digital Publishing Institute 2025
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On-line přístup:ONIX_20250220_9783725820047_69
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collection Directory of Open Access Books
description This Special Issue welcomed manuscripts that describe new compounds with antibiotic activity. Eleven papers were published, most of which describe novel compounds, including homopolymers, cyclic imides, antimicrobial peptides, nucleic acids, and derivatives of quinone, benzamidine, thiazole, and pyrazole. Two papers describe novel galenic formulations of titanate or silver nanoparticles, respectively, and one contribution describes repurposed drugs. While most of the contributions to this Special Issue describe compounds with antibacterial activity, two papers describe antimicrobial candidates that have both antibacterial and antifungal properties, and one paper describes compounds with antifungal activity.
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publishDateRange 2025
publishDateSort 2025
publisher MDPI - Multidisciplinary Digital Publishing Institute
publisherStr MDPI - Multidisciplinary Digital Publishing Institute
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spelling doab-20.500.12854ir-1527052025-02-20T12:56:31Z Molecular Methods in Antibiotics Discovery Huber, Charlotte A. antibiofilm activity candidiasis synergism synthetic peptides antifungal drugs pyrazole persisters Staphylococcus aureus Enterococcus faecalis resistance pyrrolidinone aldol antibacterial carbonic anhydrase sulfonamides inhibitors antibiotic resistance bacteria 2-aminothiazoles antifungal anticancer activity hydrazone benzimidazole sulphanilamide benzyl alkyl imidazolium ionic liquids microemulsions silver nanoparticles skin bacterial infection treatments periodontal disease periodontitis heterocyclics benzamidine bone disorders bone infections sodium titanate nanotubes anti-bacterial anti-fungal biomaterial wound infections rat model synthesis antibacterial agents quinonic-antibiotics structure–activity relationships Craig plot methicillin-resistant Staphylococcus aureus Enterococcus faecium Klebsiella pneumoniae antibacterial activity drug discovery quinone-antibiotics Free-Wilson antimicrobial bactericidal quaternary ammonium RAFT polymerization antisense oligonucleotides antisense therapies drug delivery nucleic acid engineering ribozymes riboswitches n/a thema EDItEUR::M Medicine and Nursing thema EDItEUR::M Medicine and Nursing::MB Medicine: general issues::MBN Public health and preventive medicine::MBNS Epidemiology and Medical statistics This Special Issue welcomed manuscripts that describe new compounds with antibiotic activity. Eleven papers were published, most of which describe novel compounds, including homopolymers, cyclic imides, antimicrobial peptides, nucleic acids, and derivatives of quinone, benzamidine, thiazole, and pyrazole. Two papers describe novel galenic formulations of titanate or silver nanoparticles, respectively, and one contribution describes repurposed drugs. While most of the contributions to this Special Issue describe compounds with antibacterial activity, two papers describe antimicrobial candidates that have both antibacterial and antifungal properties, and one paper describes compounds with antifungal activity. 2025-02-20T12:56:29Z 2025-02-20T12:56:29Z 2024 book ONIX_20250220_9783725820047_69 9783725820047 9783725820030 https://directory.doabooks.org/handle/20.500.12854/152705 eng application/octet-stream Attribution 4.0 International https://mdpi.com/books/pdfview/book/9820 MDPI - Multidisciplinary Digital Publishing Institute 10.3390/books978-3-7258-2003-0 10.3390/books978-3-7258-2003-0 46cabcaa-dd94-4bfe-87b4-55023c1b36d0 9783725820047 9783725820030 224 Basel open access
spellingShingle antibiofilm activity
candidiasis
synergism
synthetic peptides
antifungal drugs
pyrazole
persisters
Staphylococcus aureus
Enterococcus faecalis
resistance
pyrrolidinone
aldol
antibacterial
carbonic anhydrase
sulfonamides
inhibitors
antibiotic resistance
bacteria
2-aminothiazoles
antifungal
anticancer activity
hydrazone
benzimidazole
sulphanilamide
benzyl alkyl imidazolium ionic liquids
microemulsions
silver nanoparticles
skin bacterial infection treatments
periodontal disease
periodontitis
heterocyclics
benzamidine
bone disorders
bone infections
sodium titanate nanotubes
anti-bacterial
anti-fungal
biomaterial
wound infections
rat model
synthesis
antibacterial agents
quinonic-antibiotics
structure–activity relationships
Craig plot
methicillin-resistant Staphylococcus aureus
Enterococcus faecium
Klebsiella pneumoniae
antibacterial activity
drug discovery
quinone-antibiotics
Free-Wilson
antimicrobial
bactericidal
quaternary ammonium
RAFT polymerization
antisense oligonucleotides
antisense therapies
drug delivery
nucleic acid engineering
ribozymes
riboswitches
n/a
thema EDItEUR::M Medicine and Nursing
thema EDItEUR::M Medicine and Nursing::MB Medicine: general issues::MBN Public health and preventive medicine::MBNS Epidemiology and Medical statistics
Molecular Methods in Antibiotics Discovery
title Molecular Methods in Antibiotics Discovery
title_full Molecular Methods in Antibiotics Discovery
title_fullStr Molecular Methods in Antibiotics Discovery
title_full_unstemmed Molecular Methods in Antibiotics Discovery
title_short Molecular Methods in Antibiotics Discovery
title_sort molecular methods in antibiotics discovery
topic antibiofilm activity
candidiasis
synergism
synthetic peptides
antifungal drugs
pyrazole
persisters
Staphylococcus aureus
Enterococcus faecalis
resistance
pyrrolidinone
aldol
antibacterial
carbonic anhydrase
sulfonamides
inhibitors
antibiotic resistance
bacteria
2-aminothiazoles
antifungal
anticancer activity
hydrazone
benzimidazole
sulphanilamide
benzyl alkyl imidazolium ionic liquids
microemulsions
silver nanoparticles
skin bacterial infection treatments
periodontal disease
periodontitis
heterocyclics
benzamidine
bone disorders
bone infections
sodium titanate nanotubes
anti-bacterial
anti-fungal
biomaterial
wound infections
rat model
synthesis
antibacterial agents
quinonic-antibiotics
structure–activity relationships
Craig plot
methicillin-resistant Staphylococcus aureus
Enterococcus faecium
Klebsiella pneumoniae
antibacterial activity
drug discovery
quinone-antibiotics
Free-Wilson
antimicrobial
bactericidal
quaternary ammonium
RAFT polymerization
antisense oligonucleotides
antisense therapies
drug delivery
nucleic acid engineering
ribozymes
riboswitches
n/a
thema EDItEUR::M Medicine and Nursing
thema EDItEUR::M Medicine and Nursing::MB Medicine: general issues::MBN Public health and preventive medicine::MBNS Epidemiology and Medical statistics
topic_facet antibiofilm activity
candidiasis
synergism
synthetic peptides
antifungal drugs
pyrazole
persisters
Staphylococcus aureus
Enterococcus faecalis
resistance
pyrrolidinone
aldol
antibacterial
carbonic anhydrase
sulfonamides
inhibitors
antibiotic resistance
bacteria
2-aminothiazoles
antifungal
anticancer activity
hydrazone
benzimidazole
sulphanilamide
benzyl alkyl imidazolium ionic liquids
microemulsions
silver nanoparticles
skin bacterial infection treatments
periodontal disease
periodontitis
heterocyclics
benzamidine
bone disorders
bone infections
sodium titanate nanotubes
anti-bacterial
anti-fungal
biomaterial
wound infections
rat model
synthesis
antibacterial agents
quinonic-antibiotics
structure–activity relationships
Craig plot
methicillin-resistant Staphylococcus aureus
Enterococcus faecium
Klebsiella pneumoniae
antibacterial activity
drug discovery
quinone-antibiotics
Free-Wilson
antimicrobial
bactericidal
quaternary ammonium
RAFT polymerization
antisense oligonucleotides
antisense therapies
drug delivery
nucleic acid engineering
ribozymes
riboswitches
n/a
thema EDItEUR::M Medicine and Nursing
thema EDItEUR::M Medicine and Nursing::MB Medicine: general issues::MBN Public health and preventive medicine::MBNS Epidemiology and Medical statistics
url ONIX_20250220_9783725820047_69