Toxins in Drug Discovery and Pharmacology

Venoms from marine and terrestrial animals (cone snails, scorpions, spiders, snakes, centipedes, cnidarian, etc.) can be seen as untapped cocktails of biologically active compounds that are being increasingly recognized as a new emerging source of peptide-based therapeutics. Venomous animals are con...

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Päätekijä: Steve Peigneur (Ed.)
Aineistotyyppi: Online
Kieli:englanti
Julkaistu: MDPI - Multidisciplinary Digital Publishing Institute 2021
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Linkit:26653
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author Steve Peigneur (Ed.)
author_browse Steve Peigneur (Ed.)
author_facet Steve Peigneur (Ed.)
author_sort Steve Peigneur (Ed.)
collection Directory of Open Access Books
description Venoms from marine and terrestrial animals (cone snails, scorpions, spiders, snakes, centipedes, cnidarian, etc.) can be seen as untapped cocktails of biologically active compounds that are being increasingly recognized as a new emerging source of peptide-based therapeutics. Venomous animals are considered to be specialized predators that have evolved the most sophisticated peptide chemistry and neuropharmacology for their own biological purposes by producing venoms that contain a structural and functional diversity of neurotoxins. These neurotoxins appear to be highly selective ligands for a wide range of ion channels and receptors. Therefore, they represent interesting lead compounds for the development of analgesics, anti-cancer drugs, drugs for neurological disorders such as multiple sclerosis, Parkinson' s disease, Alzheimer' s disease, and other therapeutics. This Special Issue of Toxins aims to provide a comprehensive look at toxins and toxin-inspired leads and will focus on the mechanisms of action, structure–function relationships, and evolution of pharmacologically interesting venom components, including the most recent developments related to the emergence of venoms as an underutilized source of highly evolved bioactive peptides with clinical potential.
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spelling doab-20.500.12854ir-610712024-04-01T14:14:51Z Toxins in Drug Discovery and Pharmacology Steve Peigneur (Ed.) RA1190-1270 calcium channels acetylcholine receptors peptides botulinum toxins TRP channels spider venom peptides sodium channels opiate receptors Antibiotics cone snail venom potassium channels chloride ion channels ASIC channels NMDA receptor antimicrobial peptides thema EDItEUR::M Medicine and Nursing::MK Medical specialties, branches of medicine::MKG Pharmacology Venoms from marine and terrestrial animals (cone snails, scorpions, spiders, snakes, centipedes, cnidarian, etc.) can be seen as untapped cocktails of biologically active compounds that are being increasingly recognized as a new emerging source of peptide-based therapeutics. Venomous animals are considered to be specialized predators that have evolved the most sophisticated peptide chemistry and neuropharmacology for their own biological purposes by producing venoms that contain a structural and functional diversity of neurotoxins. These neurotoxins appear to be highly selective ligands for a wide range of ion channels and receptors. Therefore, they represent interesting lead compounds for the development of analgesics, anti-cancer drugs, drugs for neurological disorders such as multiple sclerosis, Parkinson' s disease, Alzheimer' s disease, and other therapeutics. This Special Issue of Toxins aims to provide a comprehensive look at toxins and toxin-inspired leads and will focus on the mechanisms of action, structure–function relationships, and evolution of pharmacologically interesting venom components, including the most recent developments related to the emergence of venoms as an underutilized source of highly evolved bioactive peptides with clinical potential. 2021-02-12T06:11:42Z 2021-02-12T06:11:42Z 2018-05-04 11:37:49 2018 book 26653 9783038428619 9783038428626 https://directory.doabooks.org/handle/20.500.12854/61071 eng image/png Attribution-NonCommercial-NoDerivatives 4.0 International http://www.mdpi.com/books/pdfview/book/608 http://www.mdpi.com/books/pdfview/book/608 MDPI - Multidisciplinary Digital Publishing Institute 46cabcaa-dd94-4bfe-87b4-55023c1b36d0 9783038428619 9783038428626 XII, 304 open access
spellingShingle RA1190-1270
calcium channels
acetylcholine receptors
peptides
botulinum toxins
TRP channels
spider venom peptides
sodium channels
opiate receptors
Antibiotics
cone snail venom
potassium channels
chloride ion channels
ASIC channels
NMDA receptor
antimicrobial peptides
thema EDItEUR::M Medicine and Nursing::MK Medical specialties, branches of medicine::MKG Pharmacology
Steve Peigneur (Ed.)
Toxins in Drug Discovery and Pharmacology
title Toxins in Drug Discovery and Pharmacology
title_full Toxins in Drug Discovery and Pharmacology
title_fullStr Toxins in Drug Discovery and Pharmacology
title_full_unstemmed Toxins in Drug Discovery and Pharmacology
title_short Toxins in Drug Discovery and Pharmacology
title_sort toxins in drug discovery and pharmacology
topic RA1190-1270
calcium channels
acetylcholine receptors
peptides
botulinum toxins
TRP channels
spider venom peptides
sodium channels
opiate receptors
Antibiotics
cone snail venom
potassium channels
chloride ion channels
ASIC channels
NMDA receptor
antimicrobial peptides
thema EDItEUR::M Medicine and Nursing::MK Medical specialties, branches of medicine::MKG Pharmacology
topic_facet RA1190-1270
calcium channels
acetylcholine receptors
peptides
botulinum toxins
TRP channels
spider venom peptides
sodium channels
opiate receptors
Antibiotics
cone snail venom
potassium channels
chloride ion channels
ASIC channels
NMDA receptor
antimicrobial peptides
thema EDItEUR::M Medicine and Nursing::MK Medical specialties, branches of medicine::MKG Pharmacology
url 26653
work_keys_str_mv AT stevepeigneured toxinsindrugdiscoveryandpharmacology