The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value

The book explores issues concerning the design, synthetic methods and biological evaluation of molecules of pharmaceutical interest.

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Idioma:inglês
Publicado em: MDPI - Multidisciplinary Digital Publishing Institute 2022
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collection Directory of Open Access Books
description The book explores issues concerning the design, synthetic methods and biological evaluation of molecules of pharmaceutical interest.
format Online
id doab-20.500.12854ir-76766
institution Directory of Open Access Books
language eng
publishDate 2022
publishDateRange 2022
publishDateSort 2022
publisher MDPI - Multidisciplinary Digital Publishing Institute
publisherStr MDPI - Multidisciplinary Digital Publishing Institute
record_format ojs
spelling doab-20.500.12854ir-767662024-03-28T03:32:58Z The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value Sinicropi, Maria fluorinated pyrazole aldehydes tyrosinase inhibition phosphodiesterase inhibition antibacterial activity molecular docking periodontitis SRP LDD gelcide cancer phytocomponents Tiospora cardifolia silica silver oxynitrate stability core-shell antibiofilm antimicrobial sesquiterpene inflammatory pathologies nutraceuticals triclosan surgical site infection suture abdominal surgery cost-analysis budget impact analysis spirooxindole 1,3-dipolar cycloaddition eco-friendly chemistry ROCS shape alignment lipophilicity anticancer activity sol–gel coating medical textiles antioxidant anti-inflammatory PEA derivative drug release imidazole antiproliferative antioxidant activities docking DPPH ABTS acetylcholinesterase xanthine oxidase pyrimidine-trione barbituric thiobarbituric urease inhibitors DFT N-benzylisatin-aryl hydrazones gefitinib A549 cell lines pomegranate Punica granatum L. pomegranate skin extract pomegranate fruit extract nutraceutical properties biological properties cladodes Opuntia antioxidants polyphenols SFE-CO2 rutin iso-quercitrin nicotiflorin narcissin n/a thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general thema EDItEUR::P Mathematics and Science::PN Chemistry The book explores issues concerning the design, synthetic methods and biological evaluation of molecules of pharmaceutical interest. 2022-01-11T13:41:38Z 2022-01-11T13:41:38Z 2021 book ONIX_20220111_9783036512990_501 9783036512990 9783036513003 https://directory.doabooks.org/handle/20.500.12854/76766 eng image/jpeg Attribution 4.0 International https://mdpi.com/books/pdfview/book/4215 https://mdpi.com/books/pdfview/book/4215 MDPI - Multidisciplinary Digital Publishing Institute 10.3390/books978-3-0365-1300-3 10.3390/books978-3-0365-1300-3 46cabcaa-dd94-4bfe-87b4-55023c1b36d0 9783036512990 9783036513003 218 Basel, Switzerland open access
spellingShingle fluorinated pyrazole aldehydes
tyrosinase inhibition
phosphodiesterase inhibition
antibacterial activity
molecular docking
periodontitis
SRP
LDD
gelcide
cancer
phytocomponents
Tiospora cardifolia
silica
silver oxynitrate
stability
core-shell
antibiofilm
antimicrobial
sesquiterpene
inflammatory pathologies
nutraceuticals
triclosan
surgical site infection
suture
abdominal surgery
cost-analysis
budget impact analysis
spirooxindole
1,3-dipolar cycloaddition
eco-friendly chemistry
ROCS
shape alignment
lipophilicity
anticancer activity
sol–gel coating
medical textiles
antioxidant
anti-inflammatory
PEA derivative
drug release
imidazole
antiproliferative
antioxidant activities
docking
DPPH
ABTS
acetylcholinesterase
xanthine oxidase
pyrimidine-trione
barbituric
thiobarbituric
urease inhibitors
DFT
N-benzylisatin-aryl hydrazones
gefitinib
A549 cell lines
pomegranate
Punica granatum L.
pomegranate skin extract
pomegranate fruit extract
nutraceutical properties
biological properties
cladodes
Opuntia
antioxidants
polyphenols
SFE-CO2
rutin
iso-quercitrin
nicotiflorin
narcissin
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
title The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
title_full The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
title_fullStr The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
title_full_unstemmed The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
title_short The Design, Synthesis, and Biological Evaluation of Compounds with Medicinal Value
title_sort design synthesis and biological evaluation of compounds with medicinal value
topic fluorinated pyrazole aldehydes
tyrosinase inhibition
phosphodiesterase inhibition
antibacterial activity
molecular docking
periodontitis
SRP
LDD
gelcide
cancer
phytocomponents
Tiospora cardifolia
silica
silver oxynitrate
stability
core-shell
antibiofilm
antimicrobial
sesquiterpene
inflammatory pathologies
nutraceuticals
triclosan
surgical site infection
suture
abdominal surgery
cost-analysis
budget impact analysis
spirooxindole
1,3-dipolar cycloaddition
eco-friendly chemistry
ROCS
shape alignment
lipophilicity
anticancer activity
sol–gel coating
medical textiles
antioxidant
anti-inflammatory
PEA derivative
drug release
imidazole
antiproliferative
antioxidant activities
docking
DPPH
ABTS
acetylcholinesterase
xanthine oxidase
pyrimidine-trione
barbituric
thiobarbituric
urease inhibitors
DFT
N-benzylisatin-aryl hydrazones
gefitinib
A549 cell lines
pomegranate
Punica granatum L.
pomegranate skin extract
pomegranate fruit extract
nutraceutical properties
biological properties
cladodes
Opuntia
antioxidants
polyphenols
SFE-CO2
rutin
iso-quercitrin
nicotiflorin
narcissin
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
topic_facet fluorinated pyrazole aldehydes
tyrosinase inhibition
phosphodiesterase inhibition
antibacterial activity
molecular docking
periodontitis
SRP
LDD
gelcide
cancer
phytocomponents
Tiospora cardifolia
silica
silver oxynitrate
stability
core-shell
antibiofilm
antimicrobial
sesquiterpene
inflammatory pathologies
nutraceuticals
triclosan
surgical site infection
suture
abdominal surgery
cost-analysis
budget impact analysis
spirooxindole
1,3-dipolar cycloaddition
eco-friendly chemistry
ROCS
shape alignment
lipophilicity
anticancer activity
sol–gel coating
medical textiles
antioxidant
anti-inflammatory
PEA derivative
drug release
imidazole
antiproliferative
antioxidant activities
docking
DPPH
ABTS
acetylcholinesterase
xanthine oxidase
pyrimidine-trione
barbituric
thiobarbituric
urease inhibitors
DFT
N-benzylisatin-aryl hydrazones
gefitinib
A549 cell lines
pomegranate
Punica granatum L.
pomegranate skin extract
pomegranate fruit extract
nutraceutical properties
biological properties
cladodes
Opuntia
antioxidants
polyphenols
SFE-CO2
rutin
iso-quercitrin
nicotiflorin
narcissin
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
url ONIX_20220111_9783036512990_501