Anticancer Inhibitors

The word "cancer" is associated with at least 100 different pathologies, depending on the organ involved and the type of tumor developed. Cancer is a complex disease involving multiple pathogenetic mechanisms. Characterization of different types of cancers, which distinguishes them from healthy cell...

Full description

Saved in:
Bibliographic Details
Format: Online
Language:English
Published: MDPI - Multidisciplinary Digital Publishing Institute 2023
Subjects:
Online Access:ONIX_20230220_9783036549200_44
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1869522274540847104
collection Directory of Open Access Books
description The word "cancer" is associated with at least 100 different pathologies, depending on the organ involved and the type of tumor developed. Cancer is a complex disease involving multiple pathogenetic mechanisms. Characterization of different types of cancers, which distinguishes them from healthy cells and other cancers, allows for the identification of specific targets for each individual tumor. The principle of chemotherapy is based on interference with the mechanisms that regulate the life and proliferation of cancer cells, causing their death. In recent years, there has been continuous progress in the development of therapeutic agents against cancer, which is ongoing.The Anticancer Inhibitors Special Issue focuses on new target-based anticancer agents that inhibit a specific target involved in the suppression of various types of cancer and the control of their chemoresistance.There is a collection of research and review articles on advances in drug discovery, design, and development of new inhibitor compounds with potency against various cancer types.
format Online
id doab-20.500.12854ir-97441
institution Directory of Open Access Books
language eng
publishDate 2023
publishDateRange 2023
publishDateSort 2023
publisher MDPI - Multidisciplinary Digital Publishing Institute
publisherStr MDPI - Multidisciplinary Digital Publishing Institute
record_format ojs
spelling doab-20.500.12854ir-974412024-03-28T03:32:53Z Anticancer Inhibitors Fantacuzzi, Marialuigia Ammazzalorso, Alessandra breast cancer tamoxifen LY294002 synergism apoptosis cell cycle tea (Camellia sinensis) flowers BTFS A2780/CP70 ovarian cancer cells S phase cell cycle arrest nicotinamide phosphoribosyltransferase NAD+ biosynthesis inhibitor azacyclohexane anticancer drug drug design enthalpy effect NSCLC Cathepsin K cell proliferation cell migration cell invasion mTOR isatin-hydrazones cytotoxicity CDK2 inhibitor ATP competitive inhibitor ADME analysis receptor tyrosine kinases protein-protein interactions protein engineering directed evolution angiogenesis binding affinity agonistic activity saponins phytochemicals tea (Camellia sinensis) flower ovarian cancer autophagy ZMYND8 tumorigenesis epigenetic regulation pro-oncogenic effects tumor suppression tacrine-coumarin derivatives DNA topoisomerases I II lung carcinoma cells A549 chemotherapy prodrug drug targeting overexpressed enzymes ADC ADEPT GDEPT LEAPT PROTAC cyclin-dependent kinase cancer resistance small molecule inhibitors PROTACs statins pancreatic cancer DNA microarray pitavastatin cerivastatin simvastatin fluvastatin atorvastatin pravastatin HMG-CoA reductase inhibitors n/a thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general thema EDItEUR::P Mathematics and Science::PN Chemistry The word "cancer" is associated with at least 100 different pathologies, depending on the organ involved and the type of tumor developed. Cancer is a complex disease involving multiple pathogenetic mechanisms. Characterization of different types of cancers, which distinguishes them from healthy cells and other cancers, allows for the identification of specific targets for each individual tumor. The principle of chemotherapy is based on interference with the mechanisms that regulate the life and proliferation of cancer cells, causing their death. In recent years, there has been continuous progress in the development of therapeutic agents against cancer, which is ongoing.The Anticancer Inhibitors Special Issue focuses on new target-based anticancer agents that inhibit a specific target involved in the suppression of various types of cancer and the control of their chemoresistance.There is a collection of research and review articles on advances in drug discovery, design, and development of new inhibitor compounds with potency against various cancer types. 2023-02-20T16:44:35Z 2023-02-20T16:44:35Z 2022 book ONIX_20230220_9783036549200_44 9783036549200 9783036549194 https://directory.doabooks.org/handle/20.500.12854/97441 eng image/jpeg Attribution 4.0 International https://mdpi.com/books/pdfview/book/5981 MDPI - Multidisciplinary Digital Publishing Institute 10.3390/books978-3-0365-4919-4 10.3390/books978-3-0365-4919-4 46cabcaa-dd94-4bfe-87b4-55023c1b36d0 9783036549200 9783036549194 216 Basel open access
spellingShingle breast cancer
tamoxifen
LY294002
synergism
apoptosis
cell cycle
tea (Camellia sinensis) flowers
BTFS
A2780/CP70 ovarian cancer cells
S phase cell cycle arrest
nicotinamide phosphoribosyltransferase
NAD+ biosynthesis
inhibitor
azacyclohexane
anticancer drug
drug design
enthalpy effect
NSCLC
Cathepsin K
cell proliferation
cell migration
cell invasion
mTOR
isatin-hydrazones
cytotoxicity
CDK2 inhibitor
ATP competitive inhibitor
ADME analysis
receptor tyrosine kinases
protein-protein interactions
protein engineering
directed evolution
angiogenesis
binding affinity
agonistic activity
saponins
phytochemicals
tea (Camellia sinensis) flower
ovarian cancer
autophagy
ZMYND8
tumorigenesis
epigenetic regulation
pro-oncogenic effects
tumor suppression
tacrine-coumarin derivatives
DNA
topoisomerases I
II
lung carcinoma cells
A549
chemotherapy
prodrug
drug targeting
overexpressed enzymes
ADC
ADEPT
GDEPT
LEAPT
PROTAC
cyclin-dependent kinase
cancer
resistance
small molecule inhibitors
PROTACs
statins
pancreatic cancer
DNA microarray
pitavastatin
cerivastatin
simvastatin
fluvastatin
atorvastatin
pravastatin
HMG-CoA reductase inhibitors
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
Anticancer Inhibitors
title Anticancer Inhibitors
title_full Anticancer Inhibitors
title_fullStr Anticancer Inhibitors
title_full_unstemmed Anticancer Inhibitors
title_short Anticancer Inhibitors
title_sort anticancer inhibitors
topic breast cancer
tamoxifen
LY294002
synergism
apoptosis
cell cycle
tea (Camellia sinensis) flowers
BTFS
A2780/CP70 ovarian cancer cells
S phase cell cycle arrest
nicotinamide phosphoribosyltransferase
NAD+ biosynthesis
inhibitor
azacyclohexane
anticancer drug
drug design
enthalpy effect
NSCLC
Cathepsin K
cell proliferation
cell migration
cell invasion
mTOR
isatin-hydrazones
cytotoxicity
CDK2 inhibitor
ATP competitive inhibitor
ADME analysis
receptor tyrosine kinases
protein-protein interactions
protein engineering
directed evolution
angiogenesis
binding affinity
agonistic activity
saponins
phytochemicals
tea (Camellia sinensis) flower
ovarian cancer
autophagy
ZMYND8
tumorigenesis
epigenetic regulation
pro-oncogenic effects
tumor suppression
tacrine-coumarin derivatives
DNA
topoisomerases I
II
lung carcinoma cells
A549
chemotherapy
prodrug
drug targeting
overexpressed enzymes
ADC
ADEPT
GDEPT
LEAPT
PROTAC
cyclin-dependent kinase
cancer
resistance
small molecule inhibitors
PROTACs
statins
pancreatic cancer
DNA microarray
pitavastatin
cerivastatin
simvastatin
fluvastatin
atorvastatin
pravastatin
HMG-CoA reductase inhibitors
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
topic_facet breast cancer
tamoxifen
LY294002
synergism
apoptosis
cell cycle
tea (Camellia sinensis) flowers
BTFS
A2780/CP70 ovarian cancer cells
S phase cell cycle arrest
nicotinamide phosphoribosyltransferase
NAD+ biosynthesis
inhibitor
azacyclohexane
anticancer drug
drug design
enthalpy effect
NSCLC
Cathepsin K
cell proliferation
cell migration
cell invasion
mTOR
isatin-hydrazones
cytotoxicity
CDK2 inhibitor
ATP competitive inhibitor
ADME analysis
receptor tyrosine kinases
protein-protein interactions
protein engineering
directed evolution
angiogenesis
binding affinity
agonistic activity
saponins
phytochemicals
tea (Camellia sinensis) flower
ovarian cancer
autophagy
ZMYND8
tumorigenesis
epigenetic regulation
pro-oncogenic effects
tumor suppression
tacrine-coumarin derivatives
DNA
topoisomerases I
II
lung carcinoma cells
A549
chemotherapy
prodrug
drug targeting
overexpressed enzymes
ADC
ADEPT
GDEPT
LEAPT
PROTAC
cyclin-dependent kinase
cancer
resistance
small molecule inhibitors
PROTACs
statins
pancreatic cancer
DNA microarray
pitavastatin
cerivastatin
simvastatin
fluvastatin
atorvastatin
pravastatin
HMG-CoA reductase inhibitors
n/a
thema EDItEUR::G Reference, Information and Interdisciplinary subjects::GP Research and information: general
thema EDItEUR::P Mathematics and Science::PN Chemistry
url ONIX_20230220_9783036549200_44